Research case studies Explore a selection of reports that spotlight particular areas of research at the Crick over the past five years.
Postdoctoral clinical fellows Opportunities for postdoctoral clinicians to consolidate their research experience.
Breadcrumb Mike Blackman Blackman lab Malaria Biochemistry Laboratory : Publications Lab contentLab contentIn this section Overview Vacancies Areas of interest Publications Members Clusters of malaria parasites growing inside human red blood cells. Toggle to view hero caption PublicationsYear published (-)2014 (7) Facet Year publishedPublication typeJournal article (7)Primary research (5)Method (1)Review (1) Facet Publication typeJournalBioorganic & Medicinal Chemistry Letters (2)ACS Medicinal Chemistry Letters (1)Bio-Protocol (1)Cellular Microbiology (1)Chemistry of Heterocyclic Compounds (1)Nature Communications (1) Facet Journal Publications Displaying 1 - 7 of 7Last updated : 28 March 2024 02:10 Quinoxaline-based inhibitors of malarial protease PfSUB1 Authors (7) SS Kher M Penzo S Fulle JP Ebejer PW FinnMichael Blackman A Jirgensons Chemistry of Heterocyclic Compounds Published 1 January 2015 Crick labsMike BlackmanFull details Substrate derived peptidic α-ketoamides as inhibitors of the malarial protease PfSUB1 Authors (6) Samir S Kher Maria Penzo Simone Fulle Paul W FinnMichael Blackman Aigars Jirgensons Bioorganic & Medicinal Chemistry Letters Published 7 August 2014 Crick labsMike BlackmanFull details Rational design of the first difluorostatone-based PfSUB1 inhibitors Authors (10) Simone Giovani Maria Penzo Simone Brogi Margherita Brindisi Sandra Gemma Ettore Novellino Luisa SaviniMichael Blackman Giuseppe Campiani Stefania Butini Bioorganic & Medicinal Chemistry Letters Published 23 May 2014 Crick labsMike BlackmanFull details Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit Authors (12) K Jaudzems K Tars G Maurops N Ivdra M Otikovs J Leitans[...] I Domraceva I Mutule P TrapencierisMichael Blackman A Jirgensons ACS Medicinal Chemistry Letters Published 1 April 2014 Crick labsMike BlackmanFull details Cyclic nucleotide (cAMP and cGMP) assays and capture ELISA for quantitative analysis of Plasmodium falciparum blood-stage egress Authors (4) Fiona Hackett Christine R Collins Malcolm StrathMichael Blackman Bio-Protocol Published 5 March 2014 Crick labsMike BlackmanFull details Human red blood cell-adapted Plasmodium knowlesi parasites: a new model system for malaria research Authors (6) Christof Grüring Robert W Moon Caeul LimAnthony HolderMichael Blackman Manoj T Duraisingh Cellular Microbiology Published 9 February 2014 Crick labsTony HolderMike BlackmanFull details The malaria parasite egress protease SUB1 is a calcium-dependent redox switch subtilisin Authors (9)Chrislaine Withers-Martinez Malcolm Strath Fiona Hackett Lesley F Haire Steven A HowellPhilip Walker Evangelos Christodoulou Guy G DodsonMichael Blackman Nature Communications Published 1 January 2014 Crick labs/ facilitiesMike BlackmanStructural BiologyProteomicsFull details Share the page Share on Twitter Share on Facebook Share on LinkedIn Share on Email
Quinoxaline-based inhibitors of malarial protease PfSUB1 Authors (7) SS Kher M Penzo S Fulle JP Ebejer PW FinnMichael Blackman A Jirgensons Chemistry of Heterocyclic Compounds Published 1 January 2015 Crick labsMike BlackmanFull details
Substrate derived peptidic α-ketoamides as inhibitors of the malarial protease PfSUB1 Authors (6) Samir S Kher Maria Penzo Simone Fulle Paul W FinnMichael Blackman Aigars Jirgensons Bioorganic & Medicinal Chemistry Letters Published 7 August 2014 Crick labsMike BlackmanFull details
Rational design of the first difluorostatone-based PfSUB1 inhibitors Authors (10) Simone Giovani Maria Penzo Simone Brogi Margherita Brindisi Sandra Gemma Ettore Novellino Luisa SaviniMichael Blackman Giuseppe Campiani Stefania Butini Bioorganic & Medicinal Chemistry Letters Published 23 May 2014 Crick labsMike BlackmanFull details
Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit Authors (12) K Jaudzems K Tars G Maurops N Ivdra M Otikovs J Leitans[...] I Domraceva I Mutule P TrapencierisMichael Blackman A Jirgensons ACS Medicinal Chemistry Letters Published 1 April 2014 Crick labsMike BlackmanFull details
Cyclic nucleotide (cAMP and cGMP) assays and capture ELISA for quantitative analysis of Plasmodium falciparum blood-stage egress Authors (4) Fiona Hackett Christine R Collins Malcolm StrathMichael Blackman Bio-Protocol Published 5 March 2014 Crick labsMike BlackmanFull details
Human red blood cell-adapted Plasmodium knowlesi parasites: a new model system for malaria research Authors (6) Christof Grüring Robert W Moon Caeul LimAnthony HolderMichael Blackman Manoj T Duraisingh Cellular Microbiology Published 9 February 2014 Crick labsTony HolderMike BlackmanFull details
The malaria parasite egress protease SUB1 is a calcium-dependent redox switch subtilisin Authors (9)Chrislaine Withers-Martinez Malcolm Strath Fiona Hackett Lesley F Haire Steven A HowellPhilip Walker Evangelos Christodoulou Guy G DodsonMichael Blackman Nature Communications Published 1 January 2014 Crick labs/ facilitiesMike BlackmanStructural BiologyProteomicsFull details